Histamine agonist

Drug to increase activity at histamine receptors

A histamine agonist is a drug which causes increased activity at one or more of the four histamine receptor subtypes.

H2: Betazole and Impromidine are examples of agonists used in diagnostics to increase histamine.

H3: Betahistine is a weak Histamine1 agonist and a very strong antagonist of the Histamine3 autoreceptor. Antagonizing H3 increases histaminergic tone.

See also

  • Histamine antagonist

External links

  • Histamine+agonist at the U.S. National Library of Medicine Medical Subject Headings (MeSH)
  • MeSH list of agents 82017442
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Histamine receptor modulators
H1
Agonists
  • 2-Pyridylethylamine
  • Betahistine
  • Histamine
  • HTMT
  • L-Histidine
  • UR-AK49
Antagonists
  • Unknown/unsorted: Azanator
  • Belarizine
  • Elbanizine
  • Flotrenizine
  • GSK1004723
  • Napactadine
  • Tagorizine
  • Trelnarizine
  • Trenizine
H2
Agonists
Antagonists
H3
Agonists
Antagonists
H4
Agonists
Antagonists
See also
Receptor/signaling modulators
Monoamine metabolism modulators
Monoamine reuptake inhibitors
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Types
Classes
Enzyme
see Enzyme inhibition
Ion channel
See Ion channel modulators
Receptor &
transporter
BA/M
Adrenergic
Dopaminergic
Histaminergic
Serotonergic
AA
GABAergic
Glutamatergic
Cholinergic
Cannabinoidergic
Opioidergic
Other
Miscellaneous
  • Cofactor (see Enzyme cofactors)
  • Precursor (see Amino acids)
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